Structural, conformational, biochemical, and pharmacological study of some amides derived from...

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Page 1: Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5HT 3 receptor antagonists
Page 2: Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5HT 3 receptor antagonists
Page 3: Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5HT 3 receptor antagonists
Page 4: Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5HT 3 receptor antagonists
Page 5: Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5HT 3 receptor antagonists
Page 6: Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5HT 3 receptor antagonists
Page 7: Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5HT 3 receptor antagonists
Page 8: Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5HT 3 receptor antagonists
Page 9: Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5HT 3 receptor antagonists
Page 10: Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5HT 3 receptor antagonists
Page 11: Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5HT 3 receptor antagonists
Page 12: Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5HT 3 receptor antagonists
Page 13: Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5HT 3 receptor antagonists

An AM1 study of structure and conformational isomerism in bicyclo[3.3.1] nonane and several 3,7-diaza derivatives

An AM1 study of structure and conformational isomerism in bicyclo[3.3.1] nonane and several 3,7-diaza derivatives

Sultana N, Arayne MS and Akhtar M (2014) Synthesis, Spectroscopic and Antimicrobial Properties of 1-cyclopropyl-7-[(S,S)-2,8-diazabicyclo [4.3.0]Non-8-yl]-6-fluoro-8-methoxy-1,4-dihydro-4-oxo-3

Sultana N, Arayne MS and Akhtar M (2014) Synthesis, Spectroscopic and Antimicrobial Properties of 1-cyclopropyl-7-[(S,S)-2,8-diazabicyclo [4.3.0]Non-8-yl]-6-fluoro-8-methoxy-1,4-dihydro-4-oxo-3

2,4,6,8-tetrakis(4-flurophenyl)-3,7-diazabicyclo[3.3.1]nonan-9-one S. Natarajan, V. Sudhapriya, V. Vijayakumar, N. Shoba, J. Suresh and P.L. Nilantha Laksman, Acta Cryst., 2008, E64,

2,4,6,8-tetrakis(4-flurophenyl)-3,7-diazabicyclo[3.3.1]nonan-9-one S. Natarajan, V. Sudhapriya, V. Vijayakumar, N. Shoba, J. Suresh and P.L. Nilantha Laksman, Acta Cryst., 2008, E64,

2,4,6,8-Tetrakis(4-ethylphenyl)-3,7-diazabicyclo[3.3.1]nonan-9-one K. Rajesh, V. Vijayakumar, A. P. Safwan, Kong Wai Tan and Edward R. T. Tiekink, Acta Cryst. (2010). E66, o1316

2,4,6,8-Tetrakis(4-ethylphenyl)-3,7-diazabicyclo[3.3.1]nonan-9-one K. Rajesh, V. Vijayakumar, A. P. Safwan, Kong Wai Tan and Edward R. T. Tiekink, Acta Cryst. (2010). E66, o1316

Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5-HT3 receptor antagonists

Structural, conformational, biochemical, and pharmacological study of some amides derived from 3,7-dimethyl-3,7-diazabicyclo [3.3.1] nonan-9-amine as potential 5-HT3 receptor antagonists

SR 16435 [1-(1-(Bicyclo[3.3.1]nonan-9-yl)piperidin-4-yl)indolin-2-one], a Novel Mixed Nociceptin/Orphanin FQ/ -Opioid Receptor Partial Agonist: Analgesic and Rewarding Properties

SR 16435 [1-(1-(Bicyclo[3.3.1]nonan-9-yl)piperidin-4-yl)indolin-2-one], a Novel Mixed Nociceptin/Orphanin FQ/ -Opioid Receptor Partial Agonist: Analgesic and Rewarding Properties

Photochemistry of the azoalkanes 2,3-diazabicyclo[2.2.1]hept-2-ene and spiro[cyclopropane-7,1'-[2,3]-diazabicyclo[2.2.1]hept-2-ene]: on the questions of one-bond vs. two-bond cleavage

Photochemistry of the azoalkanes 2,3-diazabicyclo[2.2.1]hept-2-ene and spiro[cyclopropane-7,1'-[2,3]-diazabicyclo[2.2.1]hept-2-ene]: on the questions of one-bond vs. two-bond cleavage

Synthesis and structural, conformational and pharmacological study of new esters derived from 3,7-dimethyl-3,7-diazabicyclo[3.3.1]nonan-9-ol

Synthesis and structural, conformational and pharmacological study of new esters derived from 3,7-dimethyl-3,7-diazabicyclo[3.3.1]nonan-9-ol

Structural, conformational, theoretical and pharmacological study of some amides derived from 3,7-dimethyl-9-[(N-substituted)-4-chlorobenzamido]3,7-diazabicyclo[3.3.1]nonane-9-carboxamide

Structural, conformational, theoretical and pharmacological study of some amides derived from 3,7-dimethyl-9-[(N-substituted)-4-chlorobenzamido]3,7-diazabicyclo[3.3.1]nonane-9-carboxamide

Synthesis and antiproliferative properties of N3/8-disubstituted 3,8-diazabicyclo[3.2.1]octane analogues of 3,8-bis[2-(3,4,5-trimethoxyphenyl)pyridin-4-yl]methyl-piperazine

Synthesis and antiproliferative properties of N3/8-disubstituted 3,8-diazabicyclo[3.2.1]octane analogues of 3,8-bis[2-(3,4,5-trimethoxyphenyl)pyridin-4-yl]methyl-piperazine

Intermolecular condensation of ethylenediamine to 1,4-diazabicyclo(2,2,2)octane over H-ZSM-5 catalysts: Effects of Si/Al ratio and crystal size

Intermolecular condensation of ethylenediamine to 1,4-diazabicyclo(2,2,2)octane over H-ZSM-5 catalysts: Effects of Si/Al ratio and crystal size

THEORETICAL STUDY OF NUCLEOPHILIC BEHAVIOUR OF 3,4-DIOXA-7-THIACYCLOPENTA[ A]PENTALENE AND 3,7-DIOXA-4- THIA-CYCLOPENTA[A]PENTALENE USING AB INTIO AND DFT BASED REACTIVITY DESCRIPTORS

THEORETICAL STUDY OF NUCLEOPHILIC BEHAVIOUR OF 3,4-DIOXA-7-THIACYCLOPENTA[ A]PENTALENE AND 3,7-DIOXA-4- THIA-CYCLOPENTA[A]PENTALENE USING AB INTIO AND DFT BASED REACTIVITY DESCRIPTORS